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References from Structural change of retinoic-acid receptor-related orphan receptor induced by binding of inverse-agonist: Molecular dynamics and ab initio molecular orbital simulations. Local targets link to admitted publications; unresolved targets remain external evidence.
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Design, synthesis, and biological evaluation of retinoic acid-related orphan receptor γt (RORγt) agonist structure-based functionality switching approach from in house RORγt inverse agonist to RORγt agonist
10.1021/acs.jmedchem.8b01181 · 2019 · External reference
structural change to tertiary sulfonamide RORc ligands led to opposite mechanisms of action
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Unresolved reference
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Unresolved reference
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