Research graph
References from Mechanistic and thermodynamic characterization of oxathiazolones as potent and selective covalent immunoproteasome inhibitors. Local targets link to admitted publications; unresolved targets remain external evidence.
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Oxathiazolones selectively inhibit the human immunoproteasome over the constitutive proteasome
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Affinity and Selectivity Assessment of Covalent Inhibitors by Free Energy Calculations
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Unresolved reference
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Unresolved reference
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Unresolved reference
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Theoretical Studies of the Acid-Base Equilibria in a Model Active Site of the Human 20S Proteasome
10.1021/acs.jcim.0c01459 · 2021 · External reference
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Catalytic Mechanism and Covalent Inhibition of UDP- N -Acetylglucosamine Enolpyruvyl Transferase (MurA): Implications to the Design of Novel Antibacterials
10.1021/acs.jcim.9b00691 · 2019 · External reference
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