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References from MUG: A mutation overview of GPCR subfamily A17 receptors. Local targets link to admitted publications; unresolved targets remain external evidence.
10.1007/s13238-016-0263-8
10.1007/s13238-016-0263-8 · External reference
CGTP collaborators, the concise guide to pharmacology 2019/20: G protein-coupled receptors
2019 · External reference
10.1124/pharmrev.120.000011
10.1124/pharmrev.120.000011 · External reference
10.1124/pr.114.009647
10.1124/pr.114.009647 · External reference
10.1038/s41467-019-13722-0
10.1038/s41467-019-13722-0 · External reference
Mechano-dependent signaling by Latrophilin/CIRL quenches cAMP in proprioceptive neurons
10.7554/elife.28360 · 2017 · External reference
10.1016/j.neuron.2014.12.057
10.1016/j.neuron.2014.12.057 · External reference
10.1016/j.ygcen.2004.12.018
10.1016/j.ygcen.2004.12.018 · External reference
G protein-coupled receptors: structure- and function-based drug discovery
10.1038/s41392-020-00435-w · 2021 · External reference
10.1016/j.tips.2019.04.001
10.1016/j.tips.2019.04.001 · External reference
10.1124/mol.63.6.1256
10.1124/mol.63.6.1256 · External reference
10.1038/nature08144
10.1038/nature08144 · External reference
Applications of machine learning in GPCR bioactive ligand discovery
10.1016/j.sbi.2019.03.022 · 2019 · External reference
10.1038/nrd.2017.178
10.1038/nrd.2017.178 · External reference
10.1016/j.tibs.2018.11.011
10.1016/j.tibs.2018.11.011 · External reference
10.1016/j.jsps.2021.04.015
10.1016/j.jsps.2021.04.015 · External reference
10.1016/j.biotechadv.2013.08.017
10.1016/j.biotechadv.2013.08.017 · External reference
10.1002/0471250953.bi0113s39
10.1002/0471250953.bi0113s39 · External reference
10.1016/j.gendis.2015.02.005
10.1016/j.gendis.2015.02.005 · External reference
Influence of disease-causing mutations on protein structural networks
10.3389/fmolb.2020.620554 · 2020 · External reference
BIO-GATS: a tool for automated GPCR template selection through a biophysical approach for homology modeling
10.3389/fmolb.2021.617176 · 2021 · External reference
The discovery of a new antibody for BRIL-fused GPCR structure determination
10.1038/s41598-020-68355-x · 2020 · External reference
Phylogenetic analysis of 277 human G-protein-coupled receptors as a tool for the prediction of orphan receptor ligands
2002 · External reference
10.1007/s10571-018-0632-3
10.1007/s10571-018-0632-3 · External reference
10.1016/s0361-9230(01)00615-3
10.1016/s0361-9230(01)00615-3 · External reference
10.1016/0006-8993(84)90117-3
10.1016/0006-8993(84)90117-3 · External reference
10.1016/b978-0-12-803111-7.00011-7
10.1016/b978-0-12-803111-7.00011-7 · 2017 · External reference
10.1016/j.pharmthera.2017.07.002
10.1016/j.pharmthera.2017.07.002 · External reference
10.1038/s41586-020-2308-7
10.1038/s41586-020-2308-7 · External reference
Variant interpretation using population databases: lessons from gnomAD
2021 · External reference
10.1093/nar/gkaa1080
10.1093/nar/gkaa1080 · External reference
Unresolved reference
1995 · External reference
Unresolved reference
External reference
10.1111/bph.13509
10.1111/bph.13509 · External reference
10.1002/cpbi.3
10.1002/cpbi.3 · External reference
Template-based protein structure modeling
10.1007/978-1-60761-842-3_6 · 2010 · External reference
Unresolved reference
External reference
Unresolved reference
External reference
10.1110/ps.062416606
10.1110/ps.062416606 · External reference
10.1002/0471250953.bi0506s15
10.1002/0471250953.bi0506s15 · External reference
10.1093/nar/gkm290
10.1093/nar/gkm290 · External reference
Unresolved reference
External reference
Unresolved reference
External reference
10.1038/s41586-021-03828-1
10.1038/s41586-021-03828-1 · External reference
10.1093/nar/gkr703
10.1093/nar/gkr703 · External reference
10.1016/0263-7855(96)00018-5
10.1016/0263-7855(96)00018-5 · External reference
10.1016/0022-2836(87)90038-6
10.1016/0022-2836(87)90038-6 · External reference
10.1016/j.jmb.2010.09.028
10.1016/j.jmb.2010.09.028 · External reference
Comparison of pathogenicity prediction tools on somatic variants
10.1016/j.jmoldx.2020.08.007 · 2020 · External reference
10.1002/humu.22225
10.1002/humu.22225 · External reference
10.1371/journal.pone.0046688
10.1371/journal.pone.0046688 · External reference
10.1038/nmeth0410-248
10.1038/nmeth0410-248 · External reference
10.1101/gr.772403
10.1101/gr.772403 · External reference
MutaFrame - an interpretative visualization framework for deleteriousness prediction of missense variants in the human exome
10.1093/bioinformatics/btab453 · 2021 · External reference
SNAP: predict effect of non-synonymous polymorphisms on function
10.1093/nar/gkm238 · 2007 · External reference
Better prediction of functional effects for sequence variants
10.1186/1471-2164-16-s8-s1 · 2015 · External reference
10.1002/humu.21047
10.1002/humu.21047 · External reference
10.1016/j.jmb.2014.04.026
10.1016/j.jmb.2014.04.026 · External reference
10.1101/gr.176601
10.1101/gr.176601 · External reference
10.21105/joss.01686
10.21105/joss.01686 · External reference
Unresolved reference
2015 · External reference
10.1146/annurev.pharmtox.41.1.593
10.1146/annurev.pharmtox.41.1.593 · External reference
10.1016/s0888-7543(03)00009-0
10.1016/s0888-7543(03)00009-0 · External reference
10.1002/ajmg.1320540419
10.1002/ajmg.1320540419 · External reference
Dopamine D4 receptor variant in Africans, D4valine194glycine, is insensitive to dopamine and clozapine: report of a homozygous individual
10.1002/(sici)1096-8628(19960122)61:3<277::aid-ajmg14>3.0.co;2-q · 1996 · External reference
Thr164Ile polymorphism of the human beta2-adrenoceptor exhibits blunted desensitization of cardiac functional responses in vivo
10.1152/ajpheart.00324.2003 · 2003 · External reference
10.1016/s0021-9258(19)49434-9
10.1016/s0021-9258(19)49434-9 · External reference
G protein-coupled receptors: the evolution of structural insight
10.3934/biophy.2017.3.491 · 2017 · External reference
10.1002/iub.1578
10.1002/iub.1578 · External reference
10.1111/j.1476-5381.2011.01629.x
10.1111/j.1476-5381.2011.01629.x · External reference
His452Tyr polymorphism in the human 5-HT2A receptor destabilizes the signaling conformation
10.1124/mol.66.5.1293 · 2004 · External reference
Pharmacogenetic prediction of clozapine response
10.1016/s0140-6736(00)02221-2 · 2000 · External reference
A naturally occurring amino acid substitution of the human serotonin 5-HT2A receptor influences amplitude and timing of intracellular calcium mobilization
10.1046/j.1471-4159.1997.68052186.x · 1997 · External reference
Amino-terminal polymorphisms of the human beta 2-adrenergic receptor impart distinct agonist-promoted regulatory properties
10.1021/bi00198a006 · 1994 · External reference
10.1006/geno.1995.1042
10.1006/geno.1995.1042 · External reference
10.1517/14728222.9.6.1247
10.1517/14728222.9.6.1247 · External reference
10.1016/j.bbamem.2006.09.029
10.1016/j.bbamem.2006.09.029 · External reference
Pharmacogenetics of the G protein-coupled receptors
10.1007/978-1-4939-0956-8_9 · 2014 · External reference
10.1016/0022-2836(71)90324-x
10.1016/0022-2836(71)90324-x · External reference
10.1002/prot.24413
10.1002/prot.24413 · External reference
10.1146/annurev-biodatasci-011720-104428
10.1146/annurev-biodatasci-011720-104428 · External reference
Solvent accessibility of residues undergoing pathogenic variations in humans: from protein structures to protein sequences
10.3389/fmolb.2020.626363 · 2020 · External reference
10.1093/genetics/149.1.445
10.1093/genetics/149.1.445 · External reference
Solvent accessibility and purifying selection within proteins of Escherichia coli and Salmonella enterica
10.1093/oxfordjournals.molbev.a026310 · 2000 · External reference
The pattern of amino acid replacements in alpha/beta-barrels
10.1093/oxfordjournals.molbev.a004009 · 2002 · External reference
10.1093/molbev/msl086
10.1093/molbev/msl086 · External reference
Proportion of solvent-exposed amino acids in a protein and rate of protein evolution
10.1093/molbev/msm019 · 2007 · External reference
10.1093/molbev/msj048
10.1093/molbev/msj048 · External reference
10.1093/molbev/msp031
10.1093/molbev/msp031 · External reference
Structural determinants of protein evolution are context-sensitive at the residue level
10.1093/molbev/msp146 · 2009 · External reference
10.1534/genetics.111.128025
10.1534/genetics.111.128025 · External reference
Characterization of disease-associated single amino acid polymorphisms in terms of sequence and structure properties
10.1006/jmbi.2001.5255 · 2002 · External reference
10.1016/j.jmb.2007.03.069
10.1016/j.jmb.2007.03.069 · External reference
Structural and genetic analysis of protein folding and stability: current Opinion in Sturctural Biology 1993, 3:589–593
10.1016/0959-440x(93)90088-3 · 1993 · External reference
10.1002/prot.10611
10.1002/prot.10611 · External reference
10.1073/pnas.041593698
10.1073/pnas.041593698 · External reference
10.1006/jmbi.2001.5353
10.1006/jmbi.2001.5353 · External reference
MENSAdb: a thorough structural analysis of membrane protein dimers
10.1093/database/baab013 · 2021 · External reference
10.1038/81919
10.1038/81919 · External reference
10.1073/pnas.98.3.880
10.1073/pnas.98.3.880 · External reference
10.1038/72440
10.1038/72440 · External reference
10.1016/j.jmb.2005.09.084
10.1016/j.jmb.2005.09.084 · External reference
10.1038/nature11896
10.1038/nature11896 · External reference
10.1038/nature09648
10.1038/nature09648 · External reference
Glycoprotein hormone receptors: determinants in leucine-rich repeats responsible for ligand specificity
10.1093/emboj/cdg260 · 2003 · External reference
A complete assessment of dopamine receptor- ligand interactions through computational methods
10.3390/molecules24071196 · 2019 · External reference
10.1038/nrd2760
10.1038/nrd2760 · External reference
10.1016/j.neuron.2017.03.016
10.1016/j.neuron.2017.03.016 · External reference
10.1021/acs.jmedchem.8b00875
10.1021/acs.jmedchem.8b00875 · External reference
10.1111/j.1476-5381.2011.01749.x
10.1111/j.1476-5381.2011.01749.x · External reference
10.1038/nchembio.199
10.1038/nchembio.199 · External reference
10.1038/nature10361
10.1038/nature10361 · External reference
10.1016/j.bbagen.2013.08.027
10.1016/j.bbagen.2013.08.027 · External reference
10.1021/acs.jcim.0c00371
10.1021/acs.jcim.0c00371 · External reference
10.1021/acschemneuro.6b00073
10.1021/acschemneuro.6b00073 · External reference
Decoding partner specificity of opioid receptor family
2021 · External reference
10.1016/j.tips.2009.02.006
10.1016/j.tips.2009.02.006 · External reference
10.1038/s41594-021-00674-7
10.1038/s41594-021-00674-7 · External reference
10.1124/mol.106.029470
10.1124/mol.106.029470 · External reference
The effect of mutations in the DRY motif on the constitutive activity and structural instability of the histamine H(2) receptor
10.1016/s0026-895x(24)26497-x · 2000 · External reference
Constitutively active mutants of the alpha 1B-adrenergic receptor: role of highly conserved polar amino acids in receptor activation
10.1002/j.1460-2075.1996.tb00726.x · 1996 · External reference
10.1073/pnas.94.3.808
10.1073/pnas.94.3.808 · External reference
Mutation of a highly conserved aspartic acid in the beta2 adrenergic receptor: constitutive activation, structural instability, and conformational rearrangement of transmembrane segment 6
10.1124/mol.56.1.175 · 1999 · External reference
10.1074/jbc.271.41.25406
10.1074/jbc.271.41.25406 · External reference
10.1124/mol.51.2.234
10.1124/mol.51.2.234 · External reference
10.1074/jbc.273.38.24322
10.1074/jbc.273.38.24322 · External reference
Effects of mutations in the highly conserved DRY motif on binding affinity, expression, and G-protein recruitment of the human angiotensin II type-2 receptor
10.1016/s0169-328x(02)00552-1 · 2002 · External reference
10.1016/j.ygeno.2006.02.009
10.1016/j.ygeno.2006.02.009 · External reference
10.1016/s0006-291x(02)00357-1
10.1016/s0006-291x(02)00357-1 · External reference
10.1124/jpet.109.163220
10.1124/jpet.109.163220 · External reference
10.1016/j.sbi.2012.03.007
10.1016/j.sbi.2012.03.007 · External reference
Functional and clinical consequences of mutations in the FSH receptor
10.1016/s0303-7207(96)03949-4 · 1996 · External reference
Functional analyses of melanocortin-4 receptor mutations identified from patients with binge eating disorder and nonobese or obese subjects
10.1210/jc.2005-0519 · 2005 · External reference
10.1038/365649a0
10.1038/365649a0 · External reference
Diversity and prevalence of somatic mutations in the thyrotropin receptor and Gs alpha genes as a cause of toxic thyroid adenomas
1997 · External reference
10.1126/science.1232808
10.1126/science.1232808 · External reference
10.1111/febs.15841
10.1111/febs.15841 · External reference
Beta2 adrenergic receptor activation. Modulation of the proline kink in transmembrane 6 by a rotamer toggle switch
2002 · External reference
The role of cysteine 6.47 in class A GPCRs
10.1186/1472-6807-13-3 · 2013 · External reference
10.1189/jlb.2ru0614-290r
10.1189/jlb.2ru0614-290r · External reference
10.1016/j.tibs.2009.07.005
10.1016/j.tibs.2009.07.005 · External reference
An activation switch in the rhodopsin family of G protein-coupled receptors: the thyrotropin receptor
10.1074/jbc.m414678200 · 2005 · External reference
10.1038/nature19107
10.1038/nature19107 · External reference
10.1016/0014-2999(96)00247-6
10.1016/0014-2999(96)00247-6 · External reference
Structural connection between activation microswitch and allosteric sodium site in GPCR signaling
10.1016/j.str.2017.12.013 · 2018 · External reference
10.1126/science.1219218
10.1126/science.1219218 · External reference
Induced effects of sodium ions on dopaminergic G-protein coupled receptors
10.1371/journal.pcbi.1000884 · 2010 · External reference
10.1016/j.mce.2016.11.023
10.1016/j.mce.2016.11.023 · External reference
10.1016/j.pharmthera.2004.08.008
10.1016/j.pharmthera.2004.08.008 · External reference
Class A and C GPCR dimers in neurodegenerative diseases
2022 · External reference
Unresolved reference
External reference
The role of phosphorylation in D1 dopamine receptor desensitization
10.1074/jbc.m308281200 · 2004 · External reference
Unresolved reference
External reference
Structural insights and functional implications of inter-individual variability in β2-adrenergic receptor
10.1038/srep24379 · 2016 · External reference
Trace Amine-associated receptor 1 (TAAR1): molecular and clinical insights for the treatment of schizophrenia and related comorbidities
10.1021/acsptsci.2c00016 · 2022 · External reference
10.1038/nrd.2016.230
10.1038/nrd.2016.230 · External reference