Research graph
References from Rh(III)-Catalyzed C–H Activation/[3 + 2] Cycloaddition for the Synthesis of Functionalized Pyrrolo[1,2- <i>a</i> ]imidazole Derivatives. Local targets link to admitted publications; unresolved targets remain external evidence.
Discovery of potent 2-aryl-6,7-dihydro-5H-pyrrolo[1,2-a]imidazoles as WDR5-WIN-site inhibitors using fragment-based methods and structure-based design
10.1021/acs.jmedchem.8b00375 · 2018 · External reference
Antimicrobial activity of DU-6681a, a parent compound of novel oral carbapenem DZ-2640
10.1128/aac.41.6.1260 · 1997 · External reference
Pharmacology of the pyrroloimidazole, SK&F 105809-II: Antiinflammatory activity and inhibition of mediator production in vivo
10.1016/0006-2952(91)90042-4 · 1991 · External reference
Structure–property optimization of a series of imidazopyridines for visceral leishmaniasis
10.1021/acsinfecdis.3c00040 · 2023 · External reference
New serotonin 5-HT1A receptor agonists endowed with antinociceptive activity in vivo
10.1021/jm400766k · 2013 · External reference
Tetrahydroindeno[1′,2′:4,5]pyrrolo[1,2-a]imidazol-5(1H)-ones as novel neonicotinoid insecticides: Reaction selectivity and substituent effects on the activity level
10.1021/jf505281p · 2015 · External reference
Pyrrole- and dihydropyrrole-fused neonicotinoids: Design, synthesis, and insecticidal evaluation
10.1021/jf3044132 · 2013 · External reference
Cyanogramide with a New Spiro[indolinone-pyrroloimidazole] Skeleton from Actinoalloteichus cyanogriseus
10.1021/ol501523d · 2014 · External reference
Design, synthesis, and application of chiral bicyclic imidazole catalysts
10.1021/acs.accounts.2c00455 · 2022 · External reference
K2S2O8/TEMPO-Induced Cascade Oxidative Cyclization/1,2-Migration of Electron-Deficient Groups: Strategy for the Construction of 1H-Pyrrol-2(3H)-ones
10.1021/acs.orglett.8b01402 · 2018 · External reference
Cu-Catalyzed Denitrogenative Transannulation of 3-Aminoindazoles To Assemble 1-Aminoisoquinolines and 3-Aminobenzothiophenes
10.1021/acs.orglett.9b02288 · 2019 · External reference
Dynamic) Kinetic Resolution of Enamines/Imines: Enantioselective N-Heterocyclic Carbene Catalyzed [3 + 3] Annulation of Bromoenals and Enamines/Imines
10.1002/anie.201813047 · 2019 · External reference
III)-catalyzed [3 + 2] annulation/pinacol rearrangement reaction of enaminones with iodonium ylides: direct synthesis of 2-spirocyclo-pyrrol-3-ones
10.1021/acs.orglett.3c02810 · 2023 · External reference
Copper-Catalyzed Cascade Cyclization Reaction of Enamines and Electron-Deficient Terminal Alkynes: Synthesis of Polysubstituted Pyrido[1,2-a]indoles
10.1021/acs.orglett.9b03739 · 2020 · External reference
Fe(OTf)3-catalyzed annulation of α,β-unsaturated ketoxime acetates with enaminones for the synthesis of functionalized 2,4-diarylpyridines
10.1039/d3qo00685a · 2023 · External reference
Cu(II)/Iodine(III) Oxide Dimerization of Heterocyclic Ketene Aminals: Tandem TEMPO Oxidation for the Highly Selective Synthesis of Functionalized 2H-Pyrrolo[1,2-a]imidazol-7(3H)-ones
10.1021/acs.orglett.0c02689 · 2020 · External reference
Multicomponent cascade reaction of 3-formylchromones: highly selective synthesis of functionalized 9-azabicyclo[3.3.1]nonane derivatives
10.1021/acs.orglett.1c02431 · 2021 · External reference
Cycloaddition and skeleton rearrangement of heterocyclic ketene aminals with 1-diazonaphthalen-2(1H)-ones for the synthesis of functionalized 1,2,3-triazoles
10.1021/acs.orglett.4c02356 · 2024 · External reference
Rh-catalyzed C–H activation, [5 + 2] cycloaddition/oxidative cascade toward functionalized benzo[f]pyrazolo[1,3]dia-zepin-6-ones
10.1021/acs.orglett.5c02561 · 2025 · External reference
Organocatalytic diastereoselective [3 + 2] cyclization of MBH carbonates with dinucleophiles: synthesis of bicyclic imidazoline derivatives that inhibit MDM2–p53 interaction
10.1039/c9cc05916d · 2019 · External reference
A Novel Naphthyridine Derivative, 3u, Induces Necroptosis at Low Concentrations and Apoptosis at High Concentrations in Human Melanoma A375 Cells. Int
10.3390/ijms19102975 · 2018 · External reference
A novel small molecule NJH-13 induces pyroptosis via the Ca2+ driven AKT-FOXO1-GSDME signaling pathway in NSCLC
10.1016/j.jare.2025.01.028 · 2025 · External reference
Synthesis and Antibacterial Activity of Thiazolo-, Oxazolo-, and Imidazolo[3,2-a][l,8]naphthyridinecarb-oxylic Acids
10.1021/jm00169a033 · 1990 · External reference
Aza-Wittig reaction with nitriles: How carbonyl function switches from reacting to activating
10.1021/acs.orglett.8b04135 · 2019 · External reference
Multicomponent tether catalysis synthesis of highly functionalized 4-(pyridin-2-ylmethyl)-2-aminopyrroles via cascade reaction
10.1021/acs.joc.9b01814 · 2019 · External reference
Substrate-controlled three-component synthesis of diverse fused heterocycles
10.1021/acs.joc.3c00497 · 2023 · External reference
Rapid syntheses of heteroaryl-substituted imidazo[1,5-a]indole and pyrrolo[1,2-c]imidazole via aerobic C2–H functionalizations
10.1021/acs.orglett.7b03596 · 2018 · External reference
Hydroxyl-directed Rh(III)-catalyzed C–H functionalization: access to benzo[de]chromenes
10.1021/acs.orglett.3c00095 · 2023 · External reference
Cascade [3 + 2]/[4 + 2] cycloaddition of enaminones with vinylene carbonate for the synthesis of functionalized pyrrolo[2,1-a]isoquinolines
10.1021/acs.orglett.4c03638 · 2024 · External reference
Yan, S.-J. Rhodium-catalyzed synthesis of N-substituted 3-acylpyrroles from enaminones and vinylene carbonate
10.1039/d4qo01816h · 2025 · External reference
Synthesis of Aggregation-Induced Emission (AIE)-Tetraarylpyrazines via Ni(II)-Catalyzed Dimerization of 2,3-Diaryl-2H-Azirines
10.1021/acs.orglett.6c01336 · 2026 · External reference
Silver-Catalyzed [3 + 2] Annulation of 2H-Azirines and CF3-Imidoyl Sulfoxonium Ylides: Access to CF3-Substituted 1H- and 2H-Pyrroles
10.1021/acs.orglett.5c02887 · 2025 · External reference
Palladium/Silver Cocatalyzed Divergent Dimerization of 2H-Azirines for Regioselective Synthesis of Tetrasubstituted Pyrroles and Pyrimidines
10.1021/acs.orglett.3c01434 · 2023 · External reference
Selective C–C Bond Formation from Rhodium-Catalyzed C–H Activation Reaction of 2-Arylpyridines with 3-Aryl-2H-azirines
10.1039/c8sc05142a · 2019 · External reference
2H-Azirines as C–C Annulation Reagents in Cu-Catalyzed Synthesis of Furo[3,2-c]quinolone Derivatives
10.1021/acs.orglett.9b01043 · 2019 · External reference
Dynamic) Kinetic Resolution of Enamines/Imines: Enantioselective N-Heterocyclic Carbene Catalyzed [3 + 3] Annulation of Bromoenals and Enamines/Imines
10.1002/anie.201813047 · ExternalCitation · doi-reference
Pharmacology of the pyrroloimidazole, SK&F 105809-II: Antiinflammatory activity and inhibition of mediator production in vivo
10.1016/0006-2952(91)90042-4 · ExternalCitation · doi-reference
A novel small molecule NJH-13 induces pyroptosis via the Ca2+ driven AKT-FOXO1-GSDME signaling pathway in NSCLC
10.1016/j.jare.2025.01.028 · ExternalCitation · doi-reference
Design, synthesis, and application of chiral bicyclic imidazole catalysts
10.1021/acs.accounts.2c00455 · ExternalCitation · doi-reference
Discovery of potent 2-aryl-6,7-dihydro-5H-pyrrolo[1,2-a]imidazoles as WDR5-WIN-site inhibitors using fragment-based methods and structure-based design
10.1021/acs.jmedchem.8b00375 · ExternalCitation · doi-reference
Substrate-controlled three-component synthesis of diverse fused heterocycles
10.1021/acs.joc.3c00497 · ExternalCitation · doi-reference
Multicomponent tether catalysis synthesis of highly functionalized 4-(pyridin-2-ylmethyl)-2-aminopyrroles via cascade reaction
10.1021/acs.joc.9b01814 · ExternalCitation · doi-reference
Cu(II)/Iodine(III) Oxide Dimerization of Heterocyclic Ketene Aminals: Tandem TEMPO Oxidation for the Highly Selective Synthesis of Functionalized 2H-Pyrrolo[1,2-a]imidazol-7(3H)-ones
10.1021/acs.orglett.0c02689 · ExternalCitation · doi-reference
Multicomponent cascade reaction of 3-formylchromones: highly selective synthesis of functionalized 9-azabicyclo[3.3.1]nonane derivatives
10.1021/acs.orglett.1c02431 · ExternalCitation · doi-reference
Hydroxyl-directed Rh(III)-catalyzed C–H functionalization: access to benzo[de]chromenes
10.1021/acs.orglett.3c00095 · ExternalCitation · doi-reference
Palladium/Silver Cocatalyzed Divergent Dimerization of 2H-Azirines for Regioselective Synthesis of Tetrasubstituted Pyrroles and Pyrimidines
10.1021/acs.orglett.3c01434 · ExternalCitation · doi-reference
III)-catalyzed [3 + 2] annulation/pinacol rearrangement reaction of enaminones with iodonium ylides: direct synthesis of 2-spirocyclo-pyrrol-3-ones
10.1021/acs.orglett.3c02810 · ExternalCitation · doi-reference
Cycloaddition and skeleton rearrangement of heterocyclic ketene aminals with 1-diazonaphthalen-2(1H)-ones for the synthesis of functionalized 1,2,3-triazoles
10.1021/acs.orglett.4c02356 · ExternalCitation · doi-reference
Cascade [3 + 2]/[4 + 2] cycloaddition of enaminones with vinylene carbonate for the synthesis of functionalized pyrrolo[2,1-a]isoquinolines
10.1021/acs.orglett.4c03638 · ExternalCitation · doi-reference
Rh-catalyzed C–H activation, [5 + 2] cycloaddition/oxidative cascade toward functionalized benzo[f]pyrazolo[1,3]dia-zepin-6-ones
10.1021/acs.orglett.5c02561 · ExternalCitation · doi-reference
Silver-Catalyzed [3 + 2] Annulation of 2H-Azirines and CF3-Imidoyl Sulfoxonium Ylides: Access to CF3-Substituted 1H- and 2H-Pyrroles
10.1021/acs.orglett.5c02887 · ExternalCitation · doi-reference
Synthesis of Aggregation-Induced Emission (AIE)-Tetraarylpyrazines via Ni(II)-Catalyzed Dimerization of 2,3-Diaryl-2H-Azirines
10.1021/acs.orglett.6c01336 · ExternalCitation · doi-reference
Rapid syntheses of heteroaryl-substituted imidazo[1,5-a]indole and pyrrolo[1,2-c]imidazole via aerobic C2–H functionalizations
10.1021/acs.orglett.7b03596 · ExternalCitation · doi-reference
K2S2O8/TEMPO-Induced Cascade Oxidative Cyclization/1,2-Migration of Electron-Deficient Groups: Strategy for the Construction of 1H-Pyrrol-2(3H)-ones
10.1021/acs.orglett.8b01402 · ExternalCitation · doi-reference
Aza-Wittig reaction with nitriles: How carbonyl function switches from reacting to activating
10.1021/acs.orglett.8b04135 · ExternalCitation · doi-reference
2H-Azirines as C–C Annulation Reagents in Cu-Catalyzed Synthesis of Furo[3,2-c]quinolone Derivatives
10.1021/acs.orglett.9b01043 · ExternalCitation · doi-reference
Cu-Catalyzed Denitrogenative Transannulation of 3-Aminoindazoles To Assemble 1-Aminoisoquinolines and 3-Aminobenzothiophenes
10.1021/acs.orglett.9b02288 · ExternalCitation · doi-reference
Copper-Catalyzed Cascade Cyclization Reaction of Enamines and Electron-Deficient Terminal Alkynes: Synthesis of Polysubstituted Pyrido[1,2-a]indoles
10.1021/acs.orglett.9b03739 · ExternalCitation · doi-reference
Structure–property optimization of a series of imidazopyridines for visceral leishmaniasis
10.1021/acsinfecdis.3c00040 · ExternalCitation · doi-reference
Pyrrole- and dihydropyrrole-fused neonicotinoids: Design, synthesis, and insecticidal evaluation
10.1021/jf3044132 · ExternalCitation · doi-reference
Tetrahydroindeno[1′,2′:4,5]pyrrolo[1,2-a]imidazol-5(1H)-ones as novel neonicotinoid insecticides: Reaction selectivity and substituent effects on the activity level
10.1021/jf505281p · ExternalCitation · doi-reference
Synthesis and Antibacterial Activity of Thiazolo-, Oxazolo-, and Imidazolo[3,2-a][l,8]naphthyridinecarb-oxylic Acids
10.1021/jm00169a033 · ExternalCitation · doi-reference
New serotonin 5-HT1A receptor agonists endowed with antinociceptive activity in vivo
10.1021/jm400766k · ExternalCitation · doi-reference
Cyanogramide with a New Spiro[indolinone-pyrroloimidazole] Skeleton from Actinoalloteichus cyanogriseus
10.1021/ol501523d · ExternalCitation · doi-reference
Selective C–C Bond Formation from Rhodium-Catalyzed C–H Activation Reaction of 2-Arylpyridines with 3-Aryl-2H-azirines
10.1039/c8sc05142a · ExternalCitation · doi-reference
Organocatalytic diastereoselective [3 + 2] cyclization of MBH carbonates with dinucleophiles: synthesis of bicyclic imidazoline derivatives that inhibit MDM2–p53 interaction
10.1039/c9cc05916d · ExternalCitation · doi-reference
Fe(OTf)3-catalyzed annulation of α,β-unsaturated ketoxime acetates with enaminones for the synthesis of functionalized 2,4-diarylpyridines
10.1039/d3qo00685a · ExternalCitation · doi-reference
Yan, S.-J. Rhodium-catalyzed synthesis of N-substituted 3-acylpyrroles from enaminones and vinylene carbonate
10.1039/d4qo01816h · ExternalCitation · doi-reference
Antimicrobial activity of DU-6681a, a parent compound of novel oral carbapenem DZ-2640
10.1128/aac.41.6.1260 · ExternalCitation · doi-reference
A Novel Naphthyridine Derivative, 3u, Induces Necroptosis at Low Concentrations and Apoptosis at High Concentrations in Human Melanoma A375 Cells. Int
10.3390/ijms19102975 · ExternalCitation · doi-reference
