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References from Synthesis of 2,3-Disubstituted 4-Ethoxycarbonyl-β-carbolin-1-ones: Application to the Synthesis of SL651498 and Its Analogue. Local targets link to admitted publications; unresolved targets remain external evidence.
β-Carbolines from the Blue-green Alga Dichothrix Baueriana
10.1021/np50105a018 · 1994 · External reference
Novel Sponge-Derived Amino Acids. 12. Tryptophan-Derived Pigments and Accompanying Sesterterpenes from Fascaplysinopis Reticulata
10.1021/jo00010a041 · 1991 · External reference
Unresolved reference
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SL651498, a GABAA Receptor Agonist with Subtype-Selective Efficacy, as a Potential Treatment for Generalized Anxiety Disorder and Muscle Spasms
10.1111/j.1527-3458.2003.tb00241.x · 2003 · External reference
Discovery of (S)-2-Cyclopentyl-N-((1-isopropylpyrrolidin2-yl)-9-methyl-1-oxo-2,9-dihydro-1H-pyrrido[3,4-b]indole-4-carboxamide (VU0453379): A Novel, CNS Penetrant Glucagon-Like Peptide 1 Receptor (GLP-1R) Positive Allosteric Modulator (PAM)
10.1021/jm501375c · 2014 · External reference
Expeditious Access to Functionalized Tricyclic Pyrrolo-Pyridones via Tandem or Sequential C–N/C–C Bond Formations
10.1021/acs.orglett.9b03514 · 2019 · External reference
Tryptamines, Carbolines, and Related Compounds. Part II. A Convenient Synthesis of Tryptamines and β-Carbolines
10.1039/jr9560004589 · 1956 · External reference
Non-peptidic Inhibitors of Human Leukocyte Elastase. 4. Design, Synthesis, and in Vitro and in Vivo Activity of a Series of β-Carbolinone-Containing Trifluoromethyl Ketones
10.1021/jm00001a014 · 1995 · External reference
Synthesis of α-Carbolines and β-Carbolinones via Intramolecular Diels-Alder reactions of 2(1H)-Pyrazinones
10.1016/s0040-4020(98)00802-3 · 1998 · External reference
A New α-Carbolinone Synthesis Using a Rh(II)-Promoted [3 + 2]-Cycloaddition and Pd(0) Cross-Coupling/Heck Cyclization Chemistry
10.1021/ol0356338 · 2003 · External reference
3-Aryl β-Carbolin-1-Ones as a New Class of Potent Inhibitors of Tumor Cell Proliferation: Synthesis and Biological Evaluation
10.1039/b412921k · 2005 · External reference
Synthesis of Benzoindoloquinolizines via a Cu(I)-Mediated C-N Bond Formation
10.1016/j.tet.2012.01.094 · 2012 · External reference
Gold-Catalyzed Cycloisomerization of N-Propargylindole-2-carboxamides: Application toward the Synthesis of Lavendamycin Analogues
10.1021/ol801385h · 2008 · External reference
Synthesis of 4-Oxo-4,5-Dihydro-3H-Pyrrolo[2,3-c]Quinoline-1-Carboxylic Acid Ethyl Ester and Its Isomer 1-Oxo-2,9-dihydro-1H-β-carboline-4-carboxylic Acid Ethyl Ester
10.1016/s0040-4020(02)01197-3 · 2002 · External reference
Intramolecular Heck Reaction of 2- And 3-Iodoindole Derivatives for the Synthesis of β- and γ-Carbolinones
10.1016/s0040-4020(02)00688-9 · 2002 · External reference
Regioselectivity on the Palladium-Catalyzed Intramolecular Cyclization of Indole Derivatives
10.1021/jo034636v · 2003 · External reference
Intramolecular Friedel–Crafts Reaction of Indoles with Carbonyl Groups: A Simple Synthesis of 3- and 4-Substituted β-Carbolin-1-ones
10.1055/s-2008-1072613 · 2008 · External reference
Synthesis of Substituted β-Carbolines via Gold(III)-Catalyzed Cycloisomerization of N-Propargylamides β-Carbolin-1-ones
10.1016/j.tet.2009.10.033 · 2010 · External reference
Synthesis of β- and γ-Carbolinones via Pd-Catalyzed Direct Dehydrogenative Annulation (DDA) of Indole-carboxamides with Alkynes Using Air as the Oxidant
10.1021/ol1007839 · 2010 · External reference
A New, Simple, and High-Yielding Synthesis of 2,9-Dihydro-1H-pyrido[3,4-b]indol-1-ones
10.1055/s-0033-1339155 · 2014 · External reference
Reactivity of Alkynylindole-2-carboxamides in [Pd]-Catalysed C-H Activation and Phase Transfer Catalysis: Formation of Pyrrolo-diindolones vs β-Carbolinones
10.1039/c6ob00583g · 2016 · External reference
β-Carbolinone Analogues from the Ugi Silver Mine
10.1002/ejoc.201800557 · 2018 · External reference
Pd/Cu Cocatalyzed Oxidative Tandem C–H Aminocarbonylation and Dehydrogenation of Tryptamines: Synthesis of Carbolinones
10.1021/acs.joc.8b03266 · 2019 · External reference
Synthesis of Nitrogen-Containing Heterocycles Using Conjugate Addition Reactions of Nucleophiles to α,β-Unsaturated Imines
10.3987/rev-12-726 · 2012 · External reference
Synthesis of (±)-Muscopyridine Analogue Using Ring-Expansion Reaction of Cyclic β-Keto Ester via Conjugate Addition to Alkynyl Imine
10.1016/j.tet.2015.05.090 · 2015 · External reference
Synthesis of α-Carbolines Using Palladium-Catalyzed Intramolecular Amination of 3-(2-Chlorophenyl)-2-Aminopyridines
10.1002/slct.201803948 · 2019 · External reference
Domino 1,4- and 1,6-Addition Reactions of Ketene Silyl Acetals to Dialkynyl Imines Promoted by Aluminum Chloride: Synthesis of Multi-Functionalized β-Lactams
10.1021/acs.joc.9b02364 · 2019 · External reference
Formation of Dihydropyridone- and Pyridone-Based Peptide Analogs through Aza-Annulation of β-Enamino Ester and Amide Substrates with α-Amido Acrylate Derivatives
10.1021/jo9600520 · 1997 · External reference
Construction of a 3-Amino-2-pyridone Library by Ring-Closing Metathesis of α-Amino Acrylamide
10.1021/cc049939x · 2004 · External reference
A General Strategy for the Synthesis of Amino-Substituted 2-Pyridones Using a Palladium-Catalyzed Amination Reaction
10.5012/bkcs.2007.28.5.777 · 2007 · External reference
An Efficient One-Pot Synthesis of 1,4-Disubstituted 3-Amino-2-Pyridone Derivatives via Three-Component Reactions of Alkynyl Aldehydes and Amines with Ethyl 2-((Diphenylmethylene)Amino)Acetate
10.1016/j.tet.2012.03.106 · 2012 · External reference
Synthesis and Antiradical Activity of 4-Aryl(Hetaryl)-substituted 3-Aminopyridin-2(1H)-ones
10.1007/s10593-016-1809-7 · 2015 · External reference
Novel 2-Pyridone Synthesis via Nucleophilic Addition of Malonic Esters to Alkynyl Imines
10.1021/ol026283c · 2002 · External reference
Buchwald-Hartwig Reaction: An Overview
10.1016/j.jorganchem.2018.02.023 · 2018 · External reference
Synthesis of Heterocycles via Pd-Ligand Controlled Cyclization of 2-Chloro-N-(2-vinyl)aniline: Preparation of Carbazoles, Indoles, Dibenzazepines, and Acridines
10.1021/ja107511g · 2010 · External reference
Synthesis of Alkynyl(phenyl)iodonium Triflates and Their Reaction with Diethyl 2-Aminomalonate
10.1021/jo00012a025 · 1991 · External reference
Synthesis of the Pyrazolo[4,3-e][1,2,4]triazine Family of Natural Products: Nostocine A, Fluviol A and Pseudoiodinine
10.1021/ja060937l · 2006 · External reference
Copper-Catalysed Reaction of Arylacetylenes with C,N-Diarylnitrones
10.1039/c39930001107 · 1993 · External reference
Copper-Catalyzed Reaction of Terminal Alkynes with Nitrones. Selective Synthesis of 1-Aza-1-buten-3-yne and 2-Azetidinone Derivatives
10.1021/jo00121a018 · 1995 · External reference
A Novel Approach to 2-Arylated Quinolines: Electrocyclization of Alkynyl Imines via Vinylidene Complexes
10.1021/ol036190a · 2004 · External reference
An Efficient Method for the Production of Terminal Alkynes from 1,1-Dibromo-1-alkenes and its Application in the Total Synthesis of Natural Product Dihydroxerulin
10.1002/adsc.201400782 · 2015 · External reference
Highly Electron-Deficient Pyridinium-Nitrones for Rapid and Tunable Inverse-Electron-Demand Strain-Promoted Alkyne-Nitrone Cycloaddition
10.1021/acs.orglett.9b01863 · 2019 · External reference
An Asymmetric Hetero-Claisen Approach to 3-Alkyl-3-aryloxindoles
10.1021/ol901441t · 2009 · External reference
Enantioselective 1,3-Dipolar Cycloaddition of Nitrones with Ethyl Vinyl Ether: The Difference between Brønsted and Lewis Acid Catalysi
10.1002/anie.200705314 · 2008 · External reference
Enantioselective 1,3-Dipolar Cycloaddition of Nitrones with Ethyl Vinyl Ether: The Difference between Brønsted and Lewis Acid Catalysis
10.1002/anie.200705314 · 2008 · External reference
Copper-Catalyzed Synthesis of Polysubstituted Pyrroles through [3+1+1] Cycloaddition Reaction of Nitrones and Isocyanides
10.1021/acs.orglett.8b00798 · 2018 · External reference
Influence of the Side-group at C═N Bridging Bond of Bis-aryl Schiff Bases on the Wavelength of Absorption Maximum of Ultraviolet Absorption Spectra
10.1002/poc.3550 · 2016 · External reference
Gold-Catalyzed Annulation/Fragmentation: Formation of Free Gold Carbenes by Retro-Cyclopropanation
10.1021/ja104743k · 2010 · External reference
The Dual Role of 1,8-Diazabicyclo[5.4.0]undec-7-ene (DBU) in the Synthesis of Terminal Aryl- and Styryl-Acetylenes via Umpolung Reactivity
10.1021/acs.orglett.5b02398 · 2015 · External reference
