Research graph
References from Solid-Phase Synthesis of Biaryl Cyclic Lipopeptides Derived from Arylomycins. Local targets link to admitted publications; unresolved targets remain external evidence.
Cyclic Peptides Containing Biaryl and Biaryl Ether Linkages
10.1007/s10989-004-1723-1 · 2005 · External reference
Cyclic Peptide Therapeutics: Past, Present and Future
10.1016/j.cbpa.2017.02.006 · 2017 · External reference
Arylomycins A and B, New Biaryl-Bridged Lipopeptide Antibiotics Produced by Streptomyces Sp. Tü 6075. I. Taxonomy, Fermentation, Isolation and Biological Activities
10.7164/antibiotics.55.565 · 2002 · External reference
Structural and Initial Biological Analysis of Synthetic Arylomycin A2
10.1021/ja073340u · 2007 · External reference
Synthesis and Biological Characterization of Arylomycin B Antibiotics
10.1021/np200163g · 2011 · External reference
Synthesis and Characterization of the Arylomycin Lipoglycopeptide Antibiotics and the Crystallographic Analysis of Their Complex with Signal Peptidase
10.1021/ja207318n · 2011 · External reference
Broad-spectrum Antibiotic Activity of the Arylomycin Natural Products Is Masked by Natural Target Mutations
10.1016/j.chembiol.2010.09.009 · 2010 · External reference
In Vitro Activities of Arylomycin Natural-Product Antibiotics Against Staphylococcus Epidermidis and Other Coagulase-Negative Staphylococci
10.1128/aac.01459-10 · 2011 · External reference
Latent Antibiotics and the Potential of the Arylomycins for Broad-Spectrum Antibacterial Activity
10.1039/c2md20043k · 2012 · External reference
A Putative Cro-Like Repressor Contributes to Arylomycin Resistance in Staphylococcus aureus
10.1128/aac.04597-14 · 2015 · External reference
Origins of Yersinia pestis Sensitivity to the Arylomycin Antibiotics and the Inhibition of Type I Signal Peptidase
10.1128/aac.00181-15 · 2015 · External reference
Inhibition of Protein Secretion in Escherichia coli and Sub-MIC Effects of Arylomycin Antibiotics
10.1128/aac.01253-18 · 2019 · External reference
Total Synthesis of Arylomycin A2, a Signal Peptidase I (SPase I) Inhibitor
10.1055/s-2008-1078209 · 2008 · External reference
Intramolecular Suzuki–Miyaura Reaction for the Total Synthesis of Signal Peptidase Inhibitors, Arylomycins A2 and B2
10.1002/chem.201000924 · 2010 · External reference
Initial Efforts Toward the Optimization of Arylomycins for Antibiotic Activity
10.1021/jm1016126 · 2011 · External reference
Efforts Toward Broadening the Spectrum of Arylomycin Antibiotic Activity
10.1016/j.bmcl.2013.08.026 · 2013 · External reference
Scalable Access to Arylomycins via C–H Functionalization Logic
10.1021/jacs.8b00087 · 2018 · External reference
Optimized Arylomycins Are a New Class of Gram-Negative Antibiotics
10.1038/s41586-018-0483-6 · 2018 · External reference
Macrolactamization Approaches to Arylomycin Antibiotics Core
10.1021/acs.orglett.8b03603 · 2019 · External reference
Stereocontrolled Synthesis of Arylomycin-Based Gram-Negative Antibiotic GDC-5338
10.1021/acs.orglett.9b03481 · 2019 · External reference
Synthesis of Biaryl-Bridged Cyclic Peptides via Catalytic Oxidative Cross-Coupling Reactions
10.1002/anie.201913305 · 2020 · External reference
Thirteen Decades of Peptide Synthesis: Key Developments in Solid Phase Peptide Synthesis and Amide Bond Formation Utilized in Peptide Ligation
10.1007/s00726-017-2516-0 · 2018 · External reference
Solid-Phase Synthesis of Biarylalanines via Suzuki Cross-Coupling and Intramolecular N-Acyliminium Pictet–Spengler Reactions
10.1016/j.tetlet.2005.09.080 · 2005 · External reference
Application of the Suzuki–Miyaura Cross-Coupling to Increase Antimicrobial Potency Generates Promising Novel Antibacterials
10.1016/j.bmcl.2006.12.049 · 2007 · External reference
Effectiveness of the Suzuki–Miyaura Cross-Coupling Reaction for Solid-Phase Peptide Modification
10.1021/cc700128b · 2008 · External reference
Solid-Phase Synthesis of Smac Peptidomimetics Incorporating Triazoloprolines and Biarylalanines
10.1021/co200078u · 2011 · External reference
Biaryl-Bridged Macrocyclic Peptides: Conformational Constraint via Carbogenic Fusion of Natural Amino Acid Side Chains
10.1021/jo202105v · 2012 · External reference
Synthesis of Fmoc-Protected Arylphenylalanines (Bip Derivatives) via Nonaqueous Suzuki-Miyaura Cross-Coupling Reactions
10.1021/acs.joc.6b01965 · 2016 · External reference
The Suzuki–Miyaura Cross-Coupling as a Versatile Tool for Peptide Diversification and Cyclization
10.3390/catal7030074 · 2017 · External reference
Solid-Phase Synthesis of 5-Arylhistidines via a Microwave-Assisted Suzuki–Miyaura Cross-Coupling
10.1016/j.tet.2008.08.077 · 2008 · External reference
Biaryl Peptides from 4-Iodophenylalanine by Solid-Phase Borylation and Suzuki–Miyaura Cross-Coupling
10.1002/ejoc.200901350 · 2010 · External reference
Solid-Phase Synthesis of Biaryl Cyclic Peptides by Borylation and Microwave-Assisted Intramolecular Suzuki–Miyaura Reaction
10.1016/j.tet.2011.01.084 · 2011 · External reference
Solid-Phase Synthesis of 5-Arylhistidine-Containing Peptides with Antimicrobial Activity Through a Microwave-Assisted Suzuki–Miyaura Cross-Coupling
10.1002/ejoc.201200291 · 2012 · External reference
Solid-Phase Synthesis of Biaryl Cyclic Peptides Containing a 3-Aryltyrosine
10.1002/ejoc.201200832 · 2012 · External reference
Solid-Phase Synthesis of Biaryl Cyclic Peptides Containing a Histidine-Tyrosine Linkage
10.1016/j.tet.2019.03.014 · 2019 · External reference
Solid-Phase Synthesis of Biaryl Cyclic Peptides Containing a Histidine-Phenylalanine Linkage
10.1007/s10989-019-09877-5 · 2020 · External reference
Efficient Synthesis of a Phosphinate Bis-Amino Acid and Its Use in the Construction of Amphiphilic Peptides
10.1021/jo00094a036 · 1994 · External reference
Use of the SPhos Ligand to Suppress Racemization in Arylpinacolboronate Ester Suzuki Couplings Involving α-Amino Acids. Synthesis of Biaryl Derivatives of 4-Hydroxyphenylglycine, Tyrosine, and Tryptophan
10.1021/jo901899w · 2009 · External reference
Selection of Boron Reagents for Suzuki–Miyaura Coupling
10.1039/c3cs60197h · 2014 · External reference
A Method for Removal of N-BOC Protecting Groups from Substrates on TFA-Sensitive Resins
10.1016/s0040-4039(98)01631-1 · 1998 · External reference
Solid Phase Synthesis of Fmoc N-Methyl Amino Acids: Application of the Fukuyama Amine Synthesis
10.1016/s0040-4039(97)01774-7 · 1997 · External reference
oNBS–SPPS: A New Method for Solid-Phase Peptide Synthesis
10.1021/ja974252k · 1998 · External reference
Orthogonal Chemistry for the Synthesis of Thiocoraline–Triostin Hybrids. Exploring their Structure–Activity Relationship
10.1021/jm4006093 · 2013 · External reference
Color Test for Detection of Free Terminal Amino Groups in the Solid-Phase Synthesis of Peptides
10.1016/0003-2697(70)90146-6 · 1970 · External reference
Detection of Secondary Amines on Solid Phase
1995 · External reference