2H-Azirines as C–C Annulation
Reagents in Cu-Catalyzed Synthesis of Furo[3,2-c]quinolone
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10.1021/acs.orglett.9b01043 · doi-reference
Selective C–C
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of 2-Arylpyridines with 3-Aryl-2H-azirines
10.1039/c8sc05142a · doi-reference
Palladium/Silver Cocatalyzed Divergent Dimerization of 2H-Azirines
for Regioselective Synthesis of Tetrasubstituted Pyrroles and Pyrimidines
10.1021/acs.orglett.3c01434 · doi-reference
Silver-Catalyzed [3
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Ylides: Access to CF3-Substituted 1H-
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10.1021/acs.orglett.5c02887 · doi-reference
Synthesis of Aggregation-Induced Emission (AIE)-Tetraarylpyrazines
via Ni(II)-Catalyzed Dimerization of 2,3-Diaryl-2H-Azirines
10.1021/acs.orglett.6c01336 · doi-reference
Yan, S.-J. Rhodium-catalyzed synthesis
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vinylene carbonate
10.1039/d4qo01816h · doi-reference
Cascade [3 + 2]/[4
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of functionalized pyrrolo[2,1-a]isoquinolines
10.1021/acs.orglett.4c03638 · doi-reference
Hydroxyl-directed Rh(III)-catalyzed
C–H functionalization:
access to benzo[de]chromenes
10.1021/acs.orglett.3c00095 · doi-reference
Rapid syntheses
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pyrrolo[1,2-c]imidazole via aerobic C2–H functionalizations
10.1021/acs.orglett.7b03596 · doi-reference
Substrate-controlled three-component
synthesis of diverse fused heterocycles
10.1021/acs.joc.3c00497 · doi-reference
Multicomponent tether catalysis synthesis of highly
functionalized 4-(pyridin-2-ylmethyl)-2-aminopyrroles via cascade
reaction
10.1021/acs.joc.9b01814 · doi-reference
Aza-Wittig reaction with nitriles: How carbonyl function
switches from reacting to activating
10.1021/acs.orglett.8b04135 · doi-reference
Synthesis
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10.1021/jm00169a033 · doi-reference
A novel small molecule NJH-13 induces
pyroptosis via the Ca2+ driven AKT-FOXO1-GSDME signaling
pathway in NSCLC
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A Novel Naphthyridine Derivative, 3u, Induces Necroptosis at Low
Concentrations and Apoptosis at High Concentrations in Human Melanoma
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Organocatalytic diastereoselective [3 + 2] cyclization
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derivatives that inhibit MDM2–p53 interaction
10.1039/c9cc05916d · doi-reference
Rh-catalyzed
C–H activation, [5 + 2] cycloaddition/oxidative cascade toward
functionalized benzo[f]pyrazolo[1,3]dia-zepin-6-ones
10.1021/acs.orglett.5c02561 · doi-reference
Cycloaddition and skeleton rearrangement of heterocyclic
ketene aminals with 1-diazonaphthalen-2(1H)-ones
for the synthesis of functionalized 1,2,3-triazoles
10.1021/acs.orglett.4c02356 · doi-reference
Multicomponent cascade
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9-azabicyclo[3.3.1]nonane derivatives
10.1021/acs.orglett.1c02431 · doi-reference
Cu(II)/Iodine(III) Oxide Dimerization of Heterocyclic
Ketene Aminals: Tandem TEMPO Oxidation for the Highly Selective Synthesis
of Functionalized 2H-Pyrrolo[1,2-a]imidazol-7(3H)-ones
10.1021/acs.orglett.0c02689 · doi-reference
Fe(OTf)3-catalyzed annulation
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with enaminones for the synthesis of functionalized 2,4-diarylpyridines
10.1039/d3qo00685a · doi-reference
Copper-Catalyzed
Cascade Cyclization Reaction of Enamines
and Electron-Deficient Terminal Alkynes: Synthesis of Polysubstituted
Pyrido[1,2-a]indoles
10.1021/acs.orglett.9b03739 · doi-reference
III)-catalyzed [3 + 2] annulation/pinacol
rearrangement reaction of enaminones with iodonium ylides: direct
synthesis of 2-spirocyclo-pyrrol-3-ones
10.1021/acs.orglett.3c02810 · doi-reference
Dynamic) Kinetic
Resolution of Enamines/Imines: Enantioselective N-Heterocyclic Carbene Catalyzed [3 + 3] Annulation of Bromoenals
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10.1002/anie.201813047 · doi-reference
Cu-Catalyzed
Denitrogenative Transannulation of 3-Aminoindazoles To Assemble 1-Aminoisoquinolines
and 3-Aminobenzothiophenes
10.1021/acs.orglett.9b02288 · doi-reference
K2S2O8/TEMPO-Induced
Cascade Oxidative Cyclization/1,2-Migration of Electron-Deficient
Groups: Strategy for the Construction of 1H-Pyrrol-2(3H)-ones
10.1021/acs.orglett.8b01402 · doi-reference
Design, synthesis,
and application
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10.1021/acs.accounts.2c00455 · doi-reference
Cyanogramide
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cyanogriseus
10.1021/ol501523d · doi-reference
Pyrrole- and dihydropyrrole-fused neonicotinoids: Design,
synthesis, and insecticidal evaluation
10.1021/jf3044132 · doi-reference
Tetrahydroindeno[1′,2′:4,5]pyrrolo[1,2-a]imidazol-5(1H)-ones as novel neonicotinoid
insecticides: Reaction selectivity and substituent effects on the
activity level
10.1021/jf505281p · doi-reference
New serotonin
5-HT1A receptor agonists endowed with antinociceptive activity
in vivo
10.1021/jm400766k · doi-reference
Structure–property
optimization of a series of imidazopyridines for visceral leishmaniasis
10.1021/acsinfecdis.3c00040 · doi-reference
Pharmacology of the
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inhibition of mediator production in vivo
10.1016/0006-2952(91)90042-4 · doi-reference
Antimicrobial
activity of DU-6681a, a parent compound of novel oral carbapenem DZ-2640
10.1128/aac.41.6.1260 · doi-reference
Discovery
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methods and structure-based design
10.1021/acs.jmedchem.8b00375 · doi-reference
